1.  AllostericRegulation of Dual Function of Thrombin. Preetpal S Sidhu. Journal of Pharmacy and Pharmacology. Accepted 2013

2.    Designing Allosteric Regulators of Thrombin. Exosite 2Features Multiple Sub-Sites That Can Be Targeted By Sulfated Small Moleculesfor Inducing Inhibition. Preetpal S. Sidhu, May A. Hamdy, Akul Y.Mehta, Qibing Zhou and Umesh R. Desai. J.Med. Chem. 2013, 56, 5059-5070.

3.   PPAR δ agonist GW0742 interacts weakly with multiple nuclearreceptors including the vitamin D receptor. Premchendar Nandhikonda,Adam Yasgar, Preetpal S Sidhu, Athena M. Baranowski, Kelly Teske, Belaynesh Feleke, Megan M.McCallum, Nina Y. Yuan, Chinedum Kevin, Daniel D. Bikle, Steven D. Ayers, PaulWebb, Ganesha Bantukallu, Anton Simeonov, Ajit Jadhav, David Maloney, Leggy A.Arnold. Biochemistry, 2013, 52, 4194-4203.

4. On Scaffold Hopping: Challenges in the Discovery of SulfatedSmall Molecules as Mimetics of Glycosaminoglycans. Preetpal S. Sidhu, Philip D.Mosier, Qibing Zhou and Umesh Desai. Bioorg.Med. Chem. Lett. 2013, 23 (1),355–359.

5.    Identification of Novel Binding Site for Allosteric Regulation of Thrombin. Preetpal S. Sidhu, May A.Hamdy Aiye Liang, Philip D. Mosier, Qibing Zhou, David H. Farrell and Umesh R.Desai. J.Med. Chem., 2012, 55 (15), 6888–6897.

6.    Rational Design of Potent, Small,Synthetic Allosteric Inhibitors of Thrombin. Preetpal S. Sidhu, Aiye Liang, Akul Y. Mehta, May A. Hamdy, Qibing Zhou and Umesh R. Desai. J. Med. Chem. 2011, 54(15), 5522-5531.

7.   First Step in Synthetic, Allosteric, Direct Inhibitors of Thrombin and Factor Xa. JensonVerghese, Aiye Liang, Preetpal S. Sidhu, Qibing Zhou, Michael Hindle, and UmeshR. Desai. Bioorg. Med. Chem. Letters, 2009, 19(15), 4126.

8.    An Efficient Synthesis of HighlyFunctionalized Benzofuran Ring in One Step. Preetpal S. Sidhu. Manuscript submitted to IJPSR.

9.    Designing Inhibitors of Thrombin and Factor XIa as Newer Anticoagulants. Preetpal S.Sidhu, Qibing Zhou and Umesh Desai. Manuscript Submitted to Bioorg. Med. Chem. Lett..

10.  Development of the first nanomolar inhibitor of theVitamin D Receptor-Coactivator interaction. Preetpal S. Sidhu, PremchendraNandhikonda, Nicholas Nassif, Megan M. McCallum, Kelly Teske, Belaynesh Feleke,Nina Y. Yuan, James M. Cook, Rakesh K. Singh, Daniel D. Bikle, Leggy A. Arnold.Submitted to J. Med.Chem.

11.  Understandingthe Mechanism of Anticancer Effect of PS121912. Manuscript in Preparation.